| 词条 | Metheptazine |
| 释义 |
| Verifiedfields = changed | verifiedrevid = 462249802 | IUPAC_name = methyl 1,2-dimethyl-4-phenylazepane-4-carboxylate | image = Metheptazine.svg | width = 180 | image2 = Metheptazine-3D-balls.png | tradename = | pregnancy_AU = | pregnancy_US = | pregnancy_category = | legal_AU = | legal_CA = | legal_UK = | legal_US = | legal_status = | routes_of_administration = | bioavailability = | protein_bound = | elimination_half-life = | excretion = | CAS_number_Ref = {{cascite|changed|??}} | CAS_number = 469-78-3 | ATC_prefix = none | ATC_suffix = | PubChem = 3047717 | DrugBank_Ref = {{drugbankcite|correct|drugbank}} | DrugBank = | ChEMBL_Ref = {{ebicite|changed|EBI}} | ChEMBL = 2104520 | ChemSpiderID_Ref = {{chemspidercite|correct|chemspider}} | ChemSpiderID = 2310051 | UNII_Ref = {{fdacite|correct|FDA}} | UNII = 93X4R66P5A | C=16 | H=23 | N=1 | O=2 | molecular_weight = 261.36 g/mol | smiles = O=C(OC)C2(c1ccccc1)CC(N(C)CCC2)C | StdInChI_Ref = {{stdinchicite|correct|chemspider}} | StdInChI = 1S/C16H23NO2/c1-13-12-16(15(18)19-3,10-7-11-17(13)2)14-8-5-4-6-9-14/h4-6,8-9,13H,7,10-12H2,1-3H3 | StdInChIKey_Ref = {{stdinchicite|correct|chemspider}} | StdInChIKey = RAAFYFKWMRWOIT-UHFFFAOYSA-N | synonyms = Metheptazine }}Metheptazine is an opioid analgesic from the phenazepine family. It was developed by American Home Products in the 1950s.[1] Metheptazine produces similar effects to other opioids, including analgesia, sedation, dizziness and nausea. Metheptazine is not listed as a controlled substance under the Controlled Substances Act 1970 in the United States.[2] The Canadian Controlled Drugs and Substances Act specifically excludes the phenazepine opioids from control. References1. ^US Patent 2740777 PROCESS FOR THE PREPARATION OF HEXAHYDRO-1,3-DIMETHYL- 4-PHENYLAZEPINE-4-CARBOXYLIC ACID, ETHYL ESTER {{Opioidergics}}{{analgesic-stub}}2. ^http://www.deadiversion.usdoj.gov/quotas/conv_factor/index.html 5 : Synthetic opioids|Azepanes|Carboxylate esters|Mu-opioid agonists|Methyl esters |
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