| 词条 | Racemorphan |
| 释义 |
| IUPAC_name = (±)-17-Methylmorphinan-3-ol | image = Racemorphan.svg | width = 250 | tradename = | pregnancy_category = | legal_AU = S9 | legal_CA = Schedule I | legal_DE = Anlage II | legal_UK = Class A | legal_UN = P I | legal_US = Schedule II | routes_of_administration = | bioavailability = | protein_bound = | metabolism = | elimination_half-life = | excretion = | CAS_number = 297-90-5 | CAS_supplemental = {{CAS|5985-35-3}} (HBr) | ATC_prefix = | ATC_suffix = | PubChem = 3918 | ChemSpiderID = 3781 | UNII_Ref = {{fdacite|correct|FDA}} | UNII = V7R79HN3XD | ChEMBL = 20803 | C=17 | H=23 | N=1 | O=1 | molecular_weight = 257.37 g/mol | StdInChI = 1S/C17H23NO/c1-18-9-8-17-7-3-2-4-14(17)16(18)10-12-5-6-13(19)11-15(12)17/h5-6,11,14,16,19H,2-4,7-10H2,1H3 | StdInChIKey = JAQUASYNZVUNQP-UHFFFAOYSA-N | smiles = CN1CCC23CCCCC2C1Cc4ccc(O)cc34 }} Racemorphan, or morphanol, is the racemic mixture of the two stereoisomers of 17-methylmorphinan-3-ol, each with differing pharmacology and effects:
Racemorphan itself is under international control per the Single Convention on Narcotic Drugs 1961 and is therefore listed as a Schedule II Narcotic controlled substance in the US Controlled Substances Act 1970; it has an ACSCN of 9733 and in 2014 it had an aggregate annual manufacturing quota of zero. [1] The salts in use are hydrobromide (free base conversion ratio 0.741), hydrochloride (0.876), and tartrate (0.632). See also
References1. ^{{cite web|url=http://www.deadiversion.usdoj.gov/quotas/conv_factor/index.html|title=Conversion Factors for Controlled Substances|author=|date=|website=www.deadiversion.usdoj.gov}} {{Hallucinogens}}{{Navboxes| title = Pharmacodynamics | titlestyle = background:#ccccff | list1 ={{Glycine receptor modulators}}{{Ion channel modulators}}{{Ionotropic glutamate receptor modulators}}{{Monoamine reuptake inhibitors}}{{Nicotinic acetylcholine receptor modulators}}{{Opioid receptor modulators}}{{Sigma receptor modulators}} }}{{nervous-system-drug-stub}}{{respiratory-system-drug-stub}} 10 : Morphinans|Opioids|Phenols|Glycine receptor antagonists|NMDA receptor antagonists|Nicotinic antagonists|Mu-opioid agonists|Serotonin-norepinephrine reuptake inhibitors|Sigma agonists|Calcium channel blockers |
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