| 词条 | CUMYL-THPINACA |
| 释义 |
| IUPAC_name = 1-(oxan-4-ylmethyl)-N-(2-phenylpropan-2-yl)indazole-3-carboxamide | image = CUMYL-THPINACA.png | tradename = | pregnancy_AU = | pregnancy_US = | pregnancy_category = | legal_AU = | legal_CA = Schedule II | legal_UK = | legal_US = | legal_status = Illegal in China and Sweden | routes_of_administration = | bioavailability = | protein_bound = | metabolism = | elimination_half-life = | excretion = | CAS_number_Ref = | CAS_number = 1400742-50-8 | ATC_prefix = | ATC_suffix = | PubChem = 86273679 | ChemSpiderID = 48057932 | smiles = O=C(NC(C)(C)C1=CC=CC=C1)C2=NN(CC3CCOCC3)C4=C2C=CC=C4 | StdInChI = 1S/C23H27N3O2/c1-23(2,18-8-4-3-5-9-18)24-22(27)21-19-10-6-7-11-20(19)26(25-21)16-17-12-14-28-15-13-17/h3-11,17H,12-16H2,1-2H3,(H,24,27) | StdInChIKey = HINCNLQQLQFMRD-UHFFFAOYSA-N | C=23 | H=27 | N=3 | O=2 | molecular_weight = 377.5 g/mol }}CUMYL-THPINACA (also known as SGT-42) is an indazole-3-carboxamide based synthetic cannabinoid.[1] CUMYL-THPINACA acts as a potent agonist for the cannabinoid receptors, with approximately 6x selectivity for CB1, having an EC50 of 0.1nM for human CB1 receptors and 0.59nM for human CB2 receptors.[2] Legal statusSweden's public health agency suggested to classify CUMYL-THPINACA as hazardous substance on November 10, 2014.[3] As of October 2015 CUMYL-THPINACA is a controlled substance in China.[4] See also
References1. ^{{cite web | url=https://www.caymanchem.com/app/template/Product.vm/catalog/17210 | title=CUMYL-THPINACA | publisher=Cayman Chemical | accessdate=11 July 2015}} {{Cannabinoids}}{{Cannabinoidergics}}{{cannabinoid-stub}}2. ^{{cite web | url=https://www.google.com/patents/WO2014167530A1 | title=Patent WO 2014167530 - Cannabinoid compounds | work=New Zealand Patent application 623626 | date=11 April 2013 | accessdate=11 July 2015 | author=Bowden|display-authors=etal}} 3. ^{{cite web | url=http://www.folkhalsomyndigheten.se/nyheter-och-press/nyhetsarkiv/2014/november/cannabinoider-foreslas-bli-klassade-som-halsofarlig-vara/ | title=Cannabinoider föreslås bli klassade som hälsofarlig vara | accessdate=11 July 2015}} 4. ^{{cite web | url=http://www.sfda.gov.cn/WS01/CL0056/130753.html | title=关于印发《非药用类麻醉药品和精神药品列管办法》的通知 | publisher=China Food and Drug Administration | date=27 September 2015 | language=Chinese | accessdate=1 October 2015}} 3 : Cannabinoids|Designer drugs|Indazolecarboxamides |
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