词条 | Etazepine |
释义 |
| IUPAC_name = 11-ethoxy-5-methyl-5,11-dihydro-6H-dibenzo[b,e]azepin-6-one | image = Etazepine.svg | CAS_number = 88124-27-0 | ATC_prefix = None | ATC_suffix = | UNII = SBC76K7XWC | PubChem = 65662 | ChEMBL = 2106559 | ChemSpiderID = 59097 | C = 17 | H = 17 | N = 1 | O = 2 | molecular_weight = 267.322 g/mol | smiles = O=C3c1c(cccc1)C(OCC)c2c(cccc2)N3C | StdInChI = 1S/C17H17NO2/c1-3-20-16-12-8-4-5-9-13(12)17(19)18(2)15-11-7-6-10-14(15)16/h4-11,16H,3H2,1-2H3 | StdInChIKey = BLGFGFHRMMDRPC-UHFFFAOYSA-N | bioavailability = | protein_bound = | metabolism = | elimination_half-life = | excretion = | pregnancy_category = | legal_status = | routes_of_administration = }}Etazepine (INN) is an anticonvulsant with a tricyclic structure which is related to the benzodiazepines, but was never marketed.[1] It appears to exert its effects via acting through the GABAergic system.[1] See also
References1. ^1 {{cite journal |vauthors=Borsini F, Volterra G, Cutrufo C, Furio M, Meli A | title = Pharmacological profile of the new anticonvulsant etazepine | journal = Arzneimittel-Forschung | volume = 39 | issue = 4 | pages = 475–9 |date=April 1989 | pmid = 2787643 | doi = | url = }} {{Anticonvulsants}}{{GABAAR PAMs}}{{Tricyclics}}{{anticonvulsant-stub}} 5 : Anticonvulsants|Dibenzazepines|Lactams|GABAA receptor positive allosteric modulators|Abandoned drugs |
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